SYNTHESIS OF NEW [1,5]-BENZODIAZEPINE DERIVATIVES CATALYZED BY VARIOUS ALIPHATIC ACIDS
نویسندگان
چکیده
منابع مشابه
Nickel-catalyzed transamidation of aliphatic amide derivatives.
Transamidation, or the conversion of one amide to another, is a long-standing challenge in organic synthesis. Although notable progress has been made in the transamidation of primary amides, the transamidation of secondary amides has remained underdeveloped, especially when considering aliphatic substrates. Herein, we report a two-step approach to achieve the transamidation of secondary aliphat...
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ژورنال
عنوان ژورنال: Al-Azhar Journal of Pharmaceutical Sciences
سال: 2013
ISSN: 2535-1958
DOI: 10.21608/ajps.2013.7099